PC54332
|
(S)-MG132 |
133407-82-6 |
MG-132 (Z-Leu-Leu-Leu-al) 是一种有效的,可逆的蛋白酶体 (proteasome) 抑制剂,IC50 为 100 nM。MG-132 有效阻断 26S 蛋白酶体复合物的蛋白水解活性。MG-132 是一种肽醛,是自噬 (autophagy) 激活剂。MG-132 还诱导凋亡 (apoptosis)。 |
PC54336
|
1-Arachidonoyl Lysophosphatidic Acid (ammonium salt) |
799268-65-8 |
Product Type|Biochemicals|Lipids|Glycerophospholipids||Product Type|Biochemicals|Receptor Pharmacology||Research Area|Cancer||Research Area|Immunology & Inflammation|Innate Immunity||Research Area|Lipid Biochemistry|Endocannabinoid/Endocannabinoid-like||Research Area|Lipid Biochemistry|Glycerophospholipids |
PC54321
|
1-Deoxynojirimycin (hydrochloride) |
73285-50-4 |
1-Deoxynojirimycin hydrochloride (Duvoglustat hydrochloride) 是一种口服有效的 α-葡萄糖苷酶 (α-glucosidase) 抑制剂。1-Deoxynojirimycin hydrochloride 抑制餐后血糖,预防糖尿病。1-Deoxynojirimycin hydrochloride 具有降血糖、减肥和抗病毒的作用。 |
PC54313
|
14,15-Leukotriene A4 methyl ester |
75290-58-3 |
Product Type|Biochemicals|Lipids|Leukotrienes||Research Area|Lipid Biochemistry |
PC54314
|
14,15-Leukotriene C4 |
75290-60-7 |
Product Type|Biochemicals|Lipids|Leukotrienes||Research Area|Immunology & Inflammation|Inflammatory Lipid Mediators|Leukotrienes||Research Area|Immunology & Inflammation|Innate Immunity||Research Area|Lipid Biochemistry|Lipoxygenase Pathways |
PC54315
|
14,15-Leukotriene D4 |
75290-64-1 |
Product Type|Biochemicals|Lipids|Leukotrienes||Research Area|Immunology & Inflammation|Inflammatory Lipid Mediators|Leukotrienes||Research Area|Immunology & Inflammation|Innate Immunity||Research Area|Lipid Biochemistry|Lipoxygenase Pathways |
PC54316
|
14,15-Leukotriene E4 |
1000852-57-2 |
Product Type|Biochemicals|Lipids|Leukotrienes||Research Area|Immunology & Inflammation|Innate Immunity||Research Area|Lipid Biochemistry|Lipoxygenase Pathways |
PC54330
|
A-803467 |
944261-79-4 |
A-803467 是一种强效、选择性的河豚毒素不敏感型 Nav1.8 钠通道阻断剂 (IC50=8 nM)。A-803467 在神经性疼痛和炎症性疼痛模型中有缓解疼痛作用。A-803467 通过与 ATP-binding cassette subfamily G member 2 (ABCG2) 转运蛋白的相互作用,增强了传统抗癌物的化疗敏感性。 |
PC54334
|
Benzisoxazole Hsp90 Inhibitor |
1012788-65-6 |
Product Type|Biochemicals|Small Molecule Inhibitors|Heat Shock Proteins||Research Area|Cancer||Research Area|Cell Biology|Cellular Chaperones |
PC54328
|
CAY10566 |
944808-88-2 |
CAY10566 是一种有效的,生物口服可利用的,选择性的硬脂酰辅酶 A 去饱和酶 1 (SCD1) 抑制剂,在小鼠和人酶测定中 IC50 分别为 4.5 和 26 nM。CAY10566 具有优异的细胞活性,可阻断 HepG2 细胞中饱和长链脂肪酸-CoAs (LCFA-CoAs) 向单不饱和 LCFA-CoAs 的转化 (IC50=7.9 nM 或 6.8 nM)。 |
PC54329
|
CAY10568 |
22913-17-3 |
Product Type|Biochemicals||Research Area|Neuroscience|Pain Research |
PC54323
|
CAY10583 |
862891-27-8 |
Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Immunology & Inflammation||Research Area|Lipid Biochemistry|Lipoxygenase Pathways |
PC54333
|
CAY10585 |
934593-90-5 |
LW6 (HIF-1α inhibitor) 是新颖的 HIF-1 抑制剂,IC50 值为 4.4 μM。LW6 降低 HIF-1α 蛋白表达,而不影响 HIF-1β 表达。 |
PC54324
|
CAY10592 |
685139-10-0 |
Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Cardiovascular System|Cardiovascular Diseases|Atherosclerosis||Research Area|Cardiovascular System|Lipids & Lipoproteins|Lipoproteins||Research Area|Endocrinology & Metabolism|Hormones & Receptors|PPARs||Research Area|Endocrinology & Metabolism|Metabolic Diseases|Diabetes||Research Area|Endocrinology & Metabolism|Metabolic Diseases|Obesity |
PC54326
|
CAY10595 |
916047-16-0 |
Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Immunology & Inflammation|Innate Immunity||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |
PC54325
|
CAY10597 |
916046-55-4 |
Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Immunology & Inflammation|Adaptive Immunity||Research Area|Immunology & Inflammation|Innate Immunity||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |
PC54338
|
Clioquinol |
130-26-7 |
Clioquinol (Iodochlorhydroxyquin) 是一种局部抗真菌药,具有抗肿瘤活性。Clioquinol 作为口服抗菌剂,可用于腹泻和皮肤感染的研究。 |
PC54318
|
ent-8-iso Prostaglandin F2α |
159812-83-6 |
Product Type|Biochemicals|Lipids|Isoprostanes||Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Lipid Biochemistry|Reactive O2/N2 Pathways||Research Area|Oxidative Stress & Reactive Species|Lipid Peroxidation |
PC54339
|
F16 |
36098-33-6 |
Application|Fluorescence||Product Type|Biochemicals|Labeling & Detection|Fluorescent Probes||Research Area|Cancer|Cell Death|Apoptosis |
PC54320
|
FTI-276 (trifluoroacetate salt) |
1217471-51-6 |
FTI-276 是一种有效的 protein farnesyl transferase (PFT) 抑制剂, 作用于恶性疟原虫和人类的 IC50 值分别为 0.9 nM 和 0.5 nM。 |