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氨溴索杂质

氨溴索杂质 相关产品(56)
货号 产品名 Cas 产品描述
PC54332 (S)-MG132 133407-82-6 MG-132 (Z-Leu-Leu-Leu-al) 是一种有效的,可逆的蛋白酶体 (proteasome) 抑制剂,IC50 为 100 nM。MG-132 有效阻断 26S 蛋白酶体复合物的蛋白水解活性。MG-132 是一种肽醛,是自噬 (autophagy) 激活剂。MG-132 还诱导凋亡 (apoptosis)。
PC54336 1-Arachidonoyl Lysophosphatidic Acid (ammonium salt) 799268-65-8 Product Type|Biochemicals|Lipids|Glycerophospholipids||Product Type|Biochemicals|Receptor Pharmacology||Research Area|Cancer||Research Area|Immunology & Inflammation|Innate Immunity||Research Area|Lipid Biochemistry|Endocannabinoid/Endocannabinoid-like||Research Area|Lipid Biochemistry|Glycerophospholipids
PC54321 1-Deoxynojirimycin (hydrochloride) 73285-50-4 1-Deoxynojirimycin hydrochloride (Duvoglustat hydrochloride) 是一种口服有效的 α-葡萄糖苷酶 (α-glucosidase) 抑制剂。1-Deoxynojirimycin hydrochloride 抑制餐后血糖,预防糖尿病。1-Deoxynojirimycin hydrochloride 具有降血糖、减肥和抗病毒的作用。
PC54313 14,15-Leukotriene A4 methyl ester 75290-58-3 Product Type|Biochemicals|Lipids|Leukotrienes||Research Area|Lipid Biochemistry
PC54314 14,15-Leukotriene C4 75290-60-7 Product Type|Biochemicals|Lipids|Leukotrienes||Research Area|Immunology & Inflammation|Inflammatory Lipid Mediators|Leukotrienes||Research Area|Immunology & Inflammation|Innate Immunity||Research Area|Lipid Biochemistry|Lipoxygenase Pathways
PC54315 14,15-Leukotriene D4 75290-64-1 Product Type|Biochemicals|Lipids|Leukotrienes||Research Area|Immunology & Inflammation|Inflammatory Lipid Mediators|Leukotrienes||Research Area|Immunology & Inflammation|Innate Immunity||Research Area|Lipid Biochemistry|Lipoxygenase Pathways
PC54316 14,15-Leukotriene E4 1000852-57-2 Product Type|Biochemicals|Lipids|Leukotrienes||Research Area|Immunology & Inflammation|Innate Immunity||Research Area|Lipid Biochemistry|Lipoxygenase Pathways
PC54330 A-803467 944261-79-4 A-803467 是一种强效、选择性的河豚毒素不敏感型 Nav1.8 钠通道阻断剂 (IC50=8 nM)。A-803467 在神经性疼痛和炎症性疼痛模型中有缓解疼痛作用。A-803467 通过与 ATP-binding cassette subfamily G member 2 (ABCG2) 转运蛋白的相互作用,增强了传统抗癌物的化疗敏感性。
PC54334 Benzisoxazole Hsp90 Inhibitor 1012788-65-6 Product Type|Biochemicals|Small Molecule Inhibitors|Heat Shock Proteins||Research Area|Cancer||Research Area|Cell Biology|Cellular Chaperones
PC54328 CAY10566 944808-88-2 CAY10566 是一种有效的,生物口服可利用的,选择性的硬脂酰辅酶 A 去饱和酶 1 (SCD1) 抑制剂,在小鼠和人酶测定中 IC50 分别为 4.5 和 26 nM。CAY10566 具有优异的细胞活性,可阻断 HepG2 细胞中饱和长链脂肪酸-CoAs (LCFA-CoAs) 向单不饱和 LCFA-CoAs 的转化 (IC50=7.9 nM 或 6.8 nM)。
PC54329 CAY10568 22913-17-3 Product Type|Biochemicals||Research Area|Neuroscience|Pain Research
PC54323 CAY10583 862891-27-8 Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Immunology & Inflammation||Research Area|Lipid Biochemistry|Lipoxygenase Pathways
PC54333 CAY10585 934593-90-5 LW6 (HIF-1α inhibitor) 是新颖的 HIF-1 抑制剂,IC50 值为 4.4 μM。LW6 降低 HIF-1α 蛋白表达,而不影响 HIF-1β 表达。
PC54324 CAY10592 685139-10-0 Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Cardiovascular System|Cardiovascular Diseases|Atherosclerosis||Research Area|Cardiovascular System|Lipids & Lipoproteins|Lipoproteins||Research Area|Endocrinology & Metabolism|Hormones & Receptors|PPARs||Research Area|Endocrinology & Metabolism|Metabolic Diseases|Diabetes||Research Area|Endocrinology & Metabolism|Metabolic Diseases|Obesity
PC54326 CAY10595 916047-16-0 Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Immunology & Inflammation|Innate Immunity||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway
PC54325 CAY10597 916046-55-4 Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Immunology & Inflammation|Adaptive Immunity||Research Area|Immunology & Inflammation|Innate Immunity||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway
PC54338 Clioquinol 130-26-7 Clioquinol (Iodochlorhydroxyquin) 是一种局部抗真菌药,具有抗肿瘤活性。Clioquinol 作为口服抗菌剂,可用于腹泻和皮肤感染的研究。
PC54318 ent-8-iso Prostaglandin F2α 159812-83-6 Product Type|Biochemicals|Lipids|Isoprostanes||Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Lipid Biochemistry|Reactive O2/N2 Pathways||Research Area|Oxidative Stress & Reactive Species|Lipid Peroxidation
PC54339 F16 36098-33-6 Application|Fluorescence||Product Type|Biochemicals|Labeling & Detection|Fluorescent Probes||Research Area|Cancer|Cell Death|Apoptosis
PC54320 FTI-276 (trifluoroacetate salt) 1217471-51-6 FTI-276 是一种有效的 protein farnesyl transferase (PFT) 抑制剂, 作用于恶性疟原虫和人类的 IC50 值分别为 0.9 nM 和 0.5 nM。