TRPV1

TRPV1 相关产品（10）

货号	产品名	Cas	产品描述
PC11849	AMG-517	659730-32-2	TRPV1拮抗剂,AMG 517是有效的香草素受体-1 (TRPV1) 拮抗剂，IC50值为0.5 nM。
PC11864	Capsazepine	138977-28-3	TRPV1离子通道拮抗剂,Capsazepine是感觉神经元兴奋毒素的合成类似物，和TRPV1 受体拮抗剂，其中IC50 为562 nM。
PC12429	Capsiconiate(solution)	946572-73-2	TRPV1激动剂,The capsaicin receptor, also termed as transient receptor potential vanilloid type 1 (TRPV1), is an non-selective cation, calcium permeable channel. The activation of TRPV1 has been reported to contribute to the various physiological activities o
PC12425	Docosahexaenoyl Serotonin(solution)	283601-58-1	TRPV1通道抑制剂,Docosahexaenoyl Serotonin is a potent TRPV1 antagonist [1].
PC12421	Eicosapentaenoyl Serotonin(solution)	199875-71-3	TRPV1通道抑制剂,Eicosapentaenoyl Serotonin is a dual fatty acid amide hydrolase (FAAH) and TRPV1 antagonist.
PC12060	mavatrep	956274-94-5	TRPV1拮抗剂,Mavatrep是一种口服生物有效的TRPV1拮抗剂, 对hTRPV1通道具有高亲和力, 抑制TRPV1激动剂与[3H]-Resiniferatoxin结合(Ki=6.5 nM), 对CYP亚型 3A4, 1A2, 和 2D6的酶活性作用效果较低。
PC12422	Oleoyl Serotonin(solution)	1002100-44-8	TRPV1通道抑制剂,Oleoyl Serotonin is a TRPV1 antagonist with IC50 value of 2.57 μM for human TRPV1 [1].
PC12423	Palmitoyl Serotonin	212707-51-2	TRPV1通道抑制剂,Palmitoyl Serotonin is a TRPV1 antagonist with IC50 value of 0.76 μM for human TRPV1 [1].
PC11901	SB705498	501951-42-4	高效选择性TRPV1拮抗剂,SB-705498 是一种有效的，选择性的，可口服的 TRPV1 拮抗剂，pIC50 值为 7.1。
PC12424	Stearoyl Serotonin	67964-87-8	TRPV1通道抑制剂,Stearoyl Serotonin is a TRPV1 antagonist with IC50 value of 0.76 μM for human TRPV1 [1].