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达格列净杂质

达格列净杂质 相关产品(76)
货号 产品名 Cas 产品描述
PC54583 (-)-WIN 55,212-3 (mesylate) 131543-25-4 Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Neuroscience|Cannabinoid Research|CB1 & CB2 Receptors
PC54591 1,24-dihydroxy Vitamin D3 (hydrate) 93129-94-3 Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Immunology & Inflammation|Adaptive Immunity||Research Area|Immunology & Inflammation|Autoimmunity
PC54564 19(R)-hydroxy Prostaglandin B2 211185-40-9 Application|Mass Spectrometry||Product Type|Biochemicals|Analytical Standards||Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway
PC54558 2-HBA 131359-24-5 2-HBA 是一个有效的 NAD(P)H: 醌受体氧化还原酶 1 (NQO1) 诱导剂,也可以激活半胱天冬酶-3 (caspase-3) 和半胱天冬酶-10 (caspase-10)。
PC54595 5-trans Prostaglandin D2 2202725-84-4 Application|Mass Spectrometry||Product Type|Biochemicals|Analytical Standards||Product Type|Biochemicals|Lipids|Prostaglandins||Product Type|Biochemicals|Pharmaceutical Impurities||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway
PC54585 Acetildenafil 831217-01-7 Product Type|Biochemicals||Research Area
PC54562 Atpenin A5 119509-24-9 Atpenin A5 是一种有效且高度特异性的 complex II 抑制剂,IC50 为 ~10 nM,且是一种有效的 mKATP 通道激动剂和心脏保护剂。
PC54584 Bosutinib 380843-75-4 Bosutinib是一种口服Src/Abl酪氨酸激酶抑制剂,IC50分别为1.2 nM和1 nM。
PC54559 CDDO methyl ester 218600-53-4 Bardoxolone methyl (NSC 713200; RTA 402; CDDO Methyl ester) 是一种合成的三萜类化合物,具有潜在的抗肿瘤和抗炎活性,作为 Nrf2 通路的激活剂和 NF-κB 途径的抑制剂。
PC54575 CGP 36216 (hydrochloride) 1781834-71-6 Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Neuroscience
PC54570 cis-2-Decenoic Acid 15790-91-7 Product Type|Biochemicals|Lipids|Fatty Acids||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Bacterial Diseases||Research Area|Infectious Disease|Fungal Diseases|Candidiasis||Research Area|Lipid Biochemistry|Fatty Acids
PC54568 CP 945,598 (hydrochloride) 686347-12-6 Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Endocrinology & Metabolism||Research Area|Neuroscience|Cannabinoid Research|CB1 & CB2 Receptors
PC54592 CPTH2 (hydrochloride) 2108899-91-6 Product Type|Biochemicals|Small Molecule Inhibitors|Acetyltransferases||Research Area|Epigenetics, Transcription, & Translation|Writers|Histone Acetylation
PC54593 Cyclosporin A 59865-13-3 Cyclosporin A (Cyclosporine A) 是一种免疫抑制剂,能与亲环素结合,抑制 calcineurin 活性的IC50 值为 7 nM。Cyclosporin A 也抑制 CD11a/CD18 粘附分子。
PC54572 Fingolimod 162359-55-9 Fingolimod (FTY720 free base) 是一种 1-磷酸鞘氨醇 (sphingosine 1-phosphate,S1P) 拮抗剂,作用于 K562 和 NK 细胞,IC50 为 0.033 nM。Fingolimod 还是一种 pak1 激活剂,免疫抑制剂。
PC54586 GSK-J1 (sodium salt) 1797832-71-3 Product Type|Biochemicals|Small Molecule Inhibitors|Demethylases||Research Area|Epigenetics, Transcription, & Translation|Erasers|Histone Demethylation||Research Area|Immunology & Inflammation|Innate Immunity
PC54587 GSK-J2 (sodium salt) 2108665-15-0 Product Type|Biochemicals|Small Molecule Inhibitors|Demethylases||Product Type|Biochemicals|Small Molecule Inhibitors|Negative Controls||Research Area|Epigenetics, Transcription, & Translation|Erasers|Histone Demethylation||Research Area|Immunology & Inflammation|Innate Immunity
PC54589 GSK-J4 (hydrochloride) 1797983-09-5 GSK-J4 hydrochloride 是一种有效的 H3K27me3/me2 去甲基化酶 JMJD3/KDM6B 和 UTX/KDM6A 双抑制剂,IC50 分别为 8.6 μM 和 6.6 μM。GSK-J4 hydrochloride 抑制 LPS 诱导的人原代巨噬细胞产生 TNF-α,IC50 值为 9 μM。GSK-J4 hydrochloride 是 GSK-J1 的细胞通透性前药。
PC54590 GSK-J5 (hydrochloride) 1797983-32-4 Product Type|Biochemicals|Small Molecule Inhibitors|Demethylases||Product Type|Biochemicals|Small Molecule Inhibitors|Negative Controls||Research Area|Epigenetics, Transcription, & Translation|Erasers|Histone Demethylation||Research Area|Immunology & Inflammation|Innate Immunity
PC54563 Hymeglusin 29066-42-0 Hymeglusin 作为一种真菌 β-内酯 antibiotic,是一种 HMG-CoA 合酶抑制剂 (IC50 = 0.12 μM)。 Hymeglusin 共价修饰酶的活性 Cys<sup>129</sup> 残基。