PC54440
|
17-DMAG |
467214-20-6 |
Product Type|Biochemicals|Small Molecule Inhibitors|Heat Shock Proteins||Research Area|Cancer||Research Area|Cell Biology|Cell Signaling|NF-κB Signaling||Research Area|Cell Biology|Cellular Chaperones||Research Area|Endocrinology & Metabolism|Metabolic Diseases|Diabetes||Research Area|Epigenetics, Transcription, & Translation|Transcription Factors||Research Area|Immunology & Inflammation||Research Area|Neuroscience |
PC54447
|
4'-O-Methylhonokiol |
68592-15-4 |
4-O-Methyl honokiol 是从厚朴中分离到的木脂素类化合物,为 PPARγ 的激动剂,可抑制 NF-κB 的活性,用于癌症,炎症等研究。 |
PC54448
|
4-Quinolone-3-Carboxamide CB2 Ligand |
1314230-69-7 |
Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Neuroscience|Cannabinoid Research|CB1 & CB2 Receptors||Research Area|Neuroscience|Pain Research |
PC54449
|
4-Quinolone-3-Carboxamide Furan CB2 Agonist |
1314230-75-5 |
Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Neuroscience|Cannabinoid Research|CB1 & CB2 Receptors||Research Area|Neuroscience|Pain Research |
PC54439
|
6-ECDCA |
459789-99-2 |
Obeticholic acid (INT-747) 是一种有效的,选择性的和口服活性的 FXR 激动剂,EC50 为 99 nM,并具有抗胆碱和抗炎作用。Obeticholic acid 还可诱导细胞自噬 (autophagy)。 |
PC54433
|
Bisdemethoxycurcumin |
33171-05-0 |
Product Type|Biochemicals|Natural Products||Research Area|Cancer||Research Area|Immunology & Inflammation|Innate Immunity|Phagocytosis||Research Area|Neuroscience|Neurodegenerative Disorders|Alzheimer’s Disease |
PC54445
|
Bisindolylmaleimide III |
137592-43-9 |
Product Type|Biochemicals|Kinase Inhibitors|PKC||Product Type|Biochemicals|Kinase Inhibitors|S6K||Product Type|Biochemicals|Small Molecule Inhibitors|Kinases||Research Area|Cell Biology|Cell Signaling |
PC54446
|
Bisindolylmaleimide XI (hydrochloride) |
145333-02-4 |
Bisindolylmaleimide XI hydrochloride (Ro 32-0432) 是一种有效、选择性和具有口服活性的 PKC 抑制剂,对 PKCα、PKCβI、PKCβII、PKCγ 的 IC50 分别为 9 nM、28 nM、31 nM、37 nM 和 108 nM。 |
PC54442
|
CAY10662 |
1184844-74-3 |
Product Type|Biochemicals|Lipids|Fatty Acids||Research Area|Cardiovascular System|Heart|Myocardial Contractility||Research Area|Lipid Biochemistry|Cytochrome P450 Pathways |
PC54443
|
CAY10665 |
1235543-17-5 |
Product Type|Biochemicals|Lipids|Fatty Acids||Research Area|Cardiovascular System|Heart|Arrhythmia||Research Area|Cardiovascular System|Heart|Myocardial Contractility||Research Area|Lipid Biochemistry|Cytochrome P450 Pathways |
PC54435
|
CAY10669 |
1243583-88-1 |
Product Type|Biochemicals|Small Molecule Inhibitors|Acetyltransferases||Research Area|Epigenetics, Transcription, & Translation|Writers|Histone Acetylation |
PC54434
|
Demethoxycurcumin |
22608-11-3 |
Product Type|Biochemicals|Natural Products||Research Area|Cancer||Research Area|Immunology & Inflammation |
PC54438
|
Dexamethasone |
50-02-2 |
Dexamethasone (Hexadecadrol) 是一种糖皮质激素受体 (glucocorticoid receptor) 激动剂。Dexamethasone 还显着降低中性粒细胞的 CD11b,CD18 和 CD62L 表达,以及单核细胞的 CD11b 和 CD18 表达。Dexamethasone 有潜力用于 COVID-19 的研究。Dexamethasone 在 LPS 诱导的巨噬细胞炎症反应中,抑制含有炎性 miRNA-155 的外泌体的产生。 |
PC54444
|
Echinomycin |
512-64-1 |
Product Type|Biochemicals|Small Molecule Inhibitors||Research Area|Cancer|Transcription Factors|HIF-1α||Research Area|Cancer|Tumor Microenvironment||Research Area|Epigenetics, Transcription, & Translation|Transcription Factors |
PC54451
|
Exendin-4 (48-86) amide (acetate) |
914454-01-6 |
Exendin-4 acetate (Exenatide acetate) 是由39个氨基酸组成的多肽。它是长效的 glucagon-like peptide-1 受体激动剂,IC50 值为 3.22 nM。 |
PC54432
|
GN25 |
1227401-27-5 |
Product Type|Biochemicals||Research Area|Cancer|Cell Signaling|p53 Signaling||Research Area|Cancer|Transcription Factors|p53 |
PC54441
|
Kendomycin |
183202-73-5 |
Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Cancer|Cell Death||Research Area|Endocrinology & Metabolism|Bone Growth & Remodeling |
PC54450
|
Palmitoyl-DL-carnitine (chloride) |
6865-14-1 |
Product Type|Biochemicals|Carnitines||Product Type|Biochemicals|Lipids|Fatty Esters/Ethers||Research Area|Cell Biology|Cell Signaling|Calcium Mobilization||Research Area|Cell Biology|ECM & Adhesion Molecules||Research Area|Cell Biology|Mitochondrial Biology||Research Area|Lipid Biochemistry|Fatty Acids|Degradation |
PC54437
|
Piperlongumine |
20069-09-4 |
Piperlongumine 是一种生物碱,具有抗炎、抗菌、抗血管生成、抗氧化、抗肿瘤和抗糖尿病等活性。在肿瘤细胞中,Piperlongumine 能够诱导 ROS 和凋亡。Piperlongumine 具有抗心肌纤维化的作用,通过抑制 ERK1/2 信号通路抑制肌成纤维细胞的转化。Piperlongumin 可用于迁移体的研究。 |
PC54452
|
Prostaglandin B1 |
13345-51-2 |
Product Type|Biochemicals|Antioxidants||Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |