PC54743
|
(R)-Butaprost |
69648-38-0 |
Product Type|Biochemicals|Lipids|Prostaglandins||Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |
PC54726
|
(±)-Clopidogrel (hydrochloride) |
130209-90-4 |
Product Type|Biochemicals||Research Area |
PC54746
|
(±)5-epi CP 55,940 |
2365471-91-4 |
Application||Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Neuroscience|Behavioral Neuroscience|Learning & Memory||Research Area|Neuroscience|Cannabinoid Research|CB1 & CB2 Receptors||Research Area|Neuroscience|Pain Research |
PC54750
|
11β-Misoprostol |
58717-36-5 |
Product Type|Biochemicals|Lipids|Prostaglandins||Product Type|Biochemicals|Pharmaceutical Impurities||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |
PC54714
|
13,14-dihydro Prostaglandin E1 |
19313-28-1 |
Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Cardiovascular System|Blood|Coagulation & Hemostasis||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |
PC54717
|
13,14-dihydro-15(R)-Prostaglandin E1 |
201848-10-4 |
Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |
PC54724
|
13,14-dihydro-15-keto Prostaglandin E1 |
5094-14-4 |
Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Cardiovascular System|Blood|Coagulation & Hemostasis||Research Area|Cardiovascular System|Cardiovascular Diseases||Research Area|Cardiovascular System|Heart||Research Area|Cardiovascular System|Vasculature|Smooth Muscle Cells||Research Area|Cardiovascular System|Vasculature|Vasodilation||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |
PC54728
|
13,14-dihydro-19(R)-hydroxy Prostaglandin E1 |
2108853-39-8 |
Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |
PC54733
|
13,14-epoxy Fluprostenol isopropyl ester |
2557327-99-6 |
Product Type|Biochemicals|Lipids|Prostaglandins||Product Type|Biochemicals|Pharmaceutical Impurities||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |
PC54740
|
15(R)-Prostaglandin E1 |
20897-91-0 |
Product Type|Biochemicals|Lipids|Prostaglandins||Product Type|Biochemicals|Small Molecule Inhibitors||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |
PC54741
|
15(S)-15-methyl Prostaglandin E1 |
35700-26-6 |
Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |
PC54734
|
15-keto Prostaglandin E1 |
22973-19-9 |
Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |
PC54745
|
16,16-dimethyl Prostaglandin E1 |
41692-15-3 |
Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Cardiovascular System|Vasculature|Vasoconstriction||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |
PC54768
|
19(R)-hydroxy Prostaglandin E1 |
64625-55-4 |
Product Type|Biochemicals|Lipids|Prostaglandins||Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Endocrinology & Metabolism|Reproductive Biology||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |
PC54772
|
6-NBDG |
108708-22-1 |
Application|Flow Cytometry||Application|Fluorescence||Product Type|Biochemicals|Labeling & Detection|Fluorescent Probes||Research Area|Endocrinology & Metabolism|Carbohydrate Metabolism||Research Area|Endocrinology & Metabolism|Metabolic Diseases|Diabetes||Research Area|Endocrinology & Metabolism|Metabolic Diseases|Metabolic Syndrome |
PC54725
|
ABT-869 |
796967-16-3 |
Linifanib (ABT-869) 是一种高效、口服的 VEGFR 和 PDGFR 家族多靶点抑制剂,对 KDR、FLT1、PDGFRβ、FLT3 的 IC50s 分别为 4、3、66、4 nM。Linifanib 具有显著的抗肿瘤活性。Linifanib 对无关 RTKs、可溶性酪氨酸激酶或丝氨酸/苏氨酸激酶的活性要低得多。Linifanib 是一种特异的 miR-10b 抑制剂,阻断 miR-10b 的生物合成。 |
PC54774
|
AD57 (hydrochloride) |
2320261-72-9 |
Product Type|Biochemicals|Kinase Inhibitors|RET||Product Type|Biochemicals|Small Molecule Inhibitors|Kinases||Research Area|Cancer|Cell Signaling|ERK/MAPK Signaling||Research Area|Cancer|Cell Signaling|SRC Family Signaling |
PC54719
|
Almorexant (hydrochloride) |
913358-93-7 |
Almorexant (ACT 078573) hydrochloride 是一种口服有效且竞争性的双 orexin receptor 拮抗剂,Kd 分别为 1.3 nM (OX1) 和 0.17 nM (OX2)。Almorexant hydrochloride 可逆地阻断食欲素-A 和食欲素-B 多肽信号。Almorexant hydrochloride 完全阻断细胞内 Ca<sup>2+</sup> 信号通路。Almorexant hydrochloride 刺激 AsPC-1 细胞 caspase-3 活性,诱导细胞凋亡 (apoptosis)。 |
PC54748
|
Axitinib |
319460-85-0 |
Axitinib是多靶点的酪氨酸激酶抑制剂,抑制 VEGFR1,VEGFR2,VEGFR3, PDGFRβ 的 IC50 值分别为 0.1, 0.2, 0.1-0.3, 1.6 nM。 |
PC54723
|
AZD 1152 (hydrochloride) |
722543-50-2 |
Product Type|Biochemicals|Kinase Inhibitors|Aurora||Product Type|Biochemicals|Small Molecule Inhibitors|Kinases||Research Area|Cancer|Cell Death|Apoptosis||Research Area|Cancer|Cell Signaling|Aurora Signaling||Research Area|Cell Biology|Cell Cycle||Research Area|Cell Biology|Cell Death|Apoptosis |