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Others 相关产品(7018

货号 产品名 中文名称 产品描述
PC17900 (+)-AS 115(solution) (+)-AS 115
PC13451 (+)-Catechin hydrate. (+)-儿茶素,儿茶酚,儿茶酸,邻苯二酚 具有各种生物活性的抗氧化类黄酮,(+)-Catechin hydrate 抑制环加氧酶-1 (COX-1) , IC50 为 1.4 μM。
PC21354 (+)-顺-地尔硫卓盐酸盐. 盐酸地尔硫卓 盐酸地尔硫卓 Diltiazem hydrochloride是钙离子流入抑制剂(缓慢通道阻断剂或钙拮抗剂)。
PC15963 (-)-Epicatechin gallate. 表儿茶素没食子酸酯 (-)-Epicatechin gallate (Epicatechin gallate) 抑制环加氧酶-1 (COX-1) , IC50 为 7.5 μM。(-)-Epicatechin gallate (Epicatechin gallate) 抑制环加氧酶-1 (COX-1) , IC50 为 7.5 μM。
PC16858 (-)-Indolactam V (-)-吲哚内酰胺V 蛋白激酶C活化剂。(-)-Indolactam V 是 PKC 的激活剂,对 η-CRD2 (PKCη 代替肽),γ-CRD2 (PKCγ 代替肽) 的 Ki 值分别为 3.36 nM 和 1.03 μM,对 PKC C1A 和 C1B 结构域的 Kd 值分别为 5.5 nM (η-C1B),7.7 nM (ε-C1B),8.3 nM (δ-C1B),18.9 nM (β-C1A-long),20.8 nM (α-C1A-long),137 nM (β-C1B),138 nM (γ-C1A) 和 213
PC10114 (-)-JQ1 (R)-(-)2-(4-(4-氯苯基)-2,3,9-三甲基-6H-噻吩并[3,2-F][1,2,4]三唑并[4,3-A][1,4]二氮杂环庚烷-6-基)乙酸叔丁酯 (-)-JQ-1 是 (+)-JQ1的异构体,可作为阴性对照物。(+)-JQ1有效 降低 BRD4 基因表达,而s (−)-JQ1 没有此作用效果
PC15008 (-)-p-Bromotetramisole Oxalate (-)-4-溴四咪唑 草酸盐 ALP抑制剂,(-)-p-Bromotetramisole Oxalate 是强效的非特异性的碱性磷酸酶抑制剂。
PC14001 (-)-槐定碱 (-)-槐定碱 Sophoridine 是一种从豆科植物槐豆斜生植物的叶子中分离出来的喹喔啉生物碱。Sophoridine 诱导细胞凋亡 (apoptosis)。Sophoridine 有可能成为胰腺癌的有效,选择性和耐受性良好的候选药物。
PC18847 (1R,3R)-3-Benzoic acid 3-carboxycyclopentyl ester (1R,3R)-3-Benzoic acid 3-carboxycyclopentyl ester
PC18800 (1R,3R)-3-Hydroxycyclopentane acetic acid methyl ester (1R,3R)-3-Hydroxycyclopentane acetic acid methyl ester
PC18848 (1R,3S)-3-Benzoic acid 3-carboxycyclopentyl ester (1R,3S)-3-Benzoic acid 3-carboxycyclopentyl ester
PC18823 (1R,3S)-3-Hydroxycyclopentane acetic acid (1R,3S)-3-Hydroxycyclopentane acetic acid
PC18809 (1R,3S)-3-Hydroxycyclopentane acetic acid methyl ester (1R,3S)-3-Hydroxycyclopentane acetic acid methyl ester
PC18836 (1R,3S)-3-Hydroxycyclopentane carboxylic acid benzyl ester (1R,3S)-3-Hydroxycyclopentane carboxylic acid benzyl ester
PC18846 (1S,3R)-3-Benzoic acid 3-carboxycyclopentyl ester (1S,3R)-3-Benzoic acid 3-carboxycyclopentyl ester
PC18822 (1S,3R)-3-Hydroxycyclopentane acetic acid (1S,3R)-3-Hydroxycyclopentane acetic acid
PC18837 (1S,3R)-3-Hydroxycyclopentane carboxylic acid benzyl ester (1S,3R)-3-Hydroxycyclopentane carboxylic acid benzyl ester
PC18821 (1S,3S)-3-Hydroxycyclopentane acetic acid (1S,3S)-3-Hydroxycyclopentane acetic acid
PC18805 (1S,3S)-3-Hydroxycyclopentane acetic acid methyl ester (1S,3S)-3-Hydroxycyclopentane acetic acid methyl ester
PC18835 (1S,3S)-3-Hydroxycyclopentane carboxylic acid benzyl ester (1S,3S)-3-Hydroxycyclopentane carboxylic acid benzyl ester