|
PC17900
|
(+)-AS 115(solution) |
|
(+)-AS 115 |
|
PC13451
|
(+)-Catechin hydrate. |
(+)-儿茶素,儿茶酚,儿茶酸,邻苯二酚 |
具有各种生物活性的抗氧化类黄酮,(+)-Catechin hydrate 抑制环加氧酶-1 (COX-1) , IC50 为 1.4 μM。 |
|
PC21354
|
(+)-顺-地尔硫卓盐酸盐. |
盐酸地尔硫卓 |
盐酸地尔硫卓 Diltiazem hydrochloride是钙离子流入抑制剂(缓慢通道阻断剂或钙拮抗剂)。 |
|
PC15963
|
(-)-Epicatechin gallate. |
表儿茶素没食子酸酯 |
(-)-Epicatechin gallate (Epicatechin gallate) 抑制环加氧酶-1 (COX-1) , IC50 为 7.5 μM。(-)-Epicatechin gallate (Epicatechin gallate) 抑制环加氧酶-1 (COX-1) , IC50 为 7.5 μM。 |
|
PC16858
|
(-)-Indolactam V |
(-)-吲哚内酰胺V |
蛋白激酶C活化剂。(-)-Indolactam V 是 PKC 的激活剂,对 η-CRD2 (PKCη 代替肽),γ-CRD2 (PKCγ 代替肽) 的 Ki 值分别为 3.36 nM 和 1.03 μM,对 PKC C1A 和 C1B 结构域的 Kd 值分别为 5.5 nM (η-C1B),7.7 nM (ε-C1B),8.3 nM (δ-C1B),18.9 nM (β-C1A-long),20.8 nM (α-C1A-long),137 nM (β-C1B),138 nM (γ-C1A) 和 213 |
|
PC10114
|
(-)-JQ1 |
(R)-(-)2-(4-(4-氯苯基)-2,3,9-三甲基-6H-噻吩并[3,2-F][1,2,4]三唑并[4,3-A][1,4]二氮杂环庚烷-6-基)乙酸叔丁酯 |
(-)-JQ-1 是 (+)-JQ1的异构体,可作为阴性对照物。(+)-JQ1有效 降低 BRD4 基因表达,而s (−)-JQ1 没有此作用效果 |
|
PC15008
|
(-)-p-Bromotetramisole Oxalate |
(-)-4-溴四咪唑 草酸盐 |
ALP抑制剂,(-)-p-Bromotetramisole Oxalate 是强效的非特异性的碱性磷酸酶抑制剂。 |
|
PC14001
|
(-)-槐定碱 |
(-)-槐定碱 |
Sophoridine 是一种从豆科植物槐豆斜生植物的叶子中分离出来的喹喔啉生物碱。Sophoridine 诱导细胞凋亡 (apoptosis)。Sophoridine 有可能成为胰腺癌的有效,选择性和耐受性良好的候选药物。 |
|
PC18847
|
(1R,3R)-3-Benzoic acid 3-carboxycyclopentyl ester |
|
(1R,3R)-3-Benzoic acid 3-carboxycyclopentyl ester |
|
PC18800
|
(1R,3R)-3-Hydroxycyclopentane acetic acid methyl ester |
|
(1R,3R)-3-Hydroxycyclopentane acetic acid methyl ester |
|
PC18848
|
(1R,3S)-3-Benzoic acid 3-carboxycyclopentyl ester |
|
(1R,3S)-3-Benzoic acid 3-carboxycyclopentyl ester |
|
PC18823
|
(1R,3S)-3-Hydroxycyclopentane acetic acid |
|
(1R,3S)-3-Hydroxycyclopentane acetic acid |
|
PC18809
|
(1R,3S)-3-Hydroxycyclopentane acetic acid methyl ester |
|
(1R,3S)-3-Hydroxycyclopentane acetic acid methyl ester |
|
PC18836
|
(1R,3S)-3-Hydroxycyclopentane carboxylic acid benzyl ester |
|
(1R,3S)-3-Hydroxycyclopentane carboxylic acid benzyl ester |
|
PC18846
|
(1S,3R)-3-Benzoic acid 3-carboxycyclopentyl ester |
|
(1S,3R)-3-Benzoic acid 3-carboxycyclopentyl ester |
|
PC18822
|
(1S,3R)-3-Hydroxycyclopentane acetic acid |
|
(1S,3R)-3-Hydroxycyclopentane acetic acid |
|
PC18837
|
(1S,3R)-3-Hydroxycyclopentane carboxylic acid benzyl ester |
|
(1S,3R)-3-Hydroxycyclopentane carboxylic acid benzyl ester |
|
PC18821
|
(1S,3S)-3-Hydroxycyclopentane acetic acid |
|
(1S,3S)-3-Hydroxycyclopentane acetic acid |
|
PC18805
|
(1S,3S)-3-Hydroxycyclopentane acetic acid methyl ester |
|
(1S,3S)-3-Hydroxycyclopentane acetic acid methyl ester |
|
PC18835
|
(1S,3S)-3-Hydroxycyclopentane carboxylic acid benzyl ester |
|
(1S,3S)-3-Hydroxycyclopentane carboxylic acid benzyl ester |