Efalizumab

目录号: PL14832 纯度: ≥98%
Efalizumab 是一种靶向 T 细胞的调节剂,是 LFA-1 α 亚基 CD11a 的人源化单克隆抗体。依法珠单抗可抑制 T 细胞激活、皮肤T细胞运输和T细胞粘附到角质形成细胞,可用于斑块银屑病研究。
CAS No. :214745-43-4
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中文名称
Efalizumab
中文别名
EFALIZUMAB ( 依法珠单抗 );依法利珠单抗
英文名称
Efalizumab
英文别名
Raptiva;Xanelim;hu 1124;Efalizumab
Cas No.
214745-43-4
包装储存
Please store the product under the recommended conditions in the Certificate of Analysis.
详情描述
Efalizumab 是一种靶向 T 细胞的调节剂,是 LFA-1 α 亚基 CD11a 的人源化单克隆抗体。依法珠单抗可抑制 T 细胞激活、皮肤T细胞运输和T细胞粘附到角质形成细胞,可用于斑块银屑病研究。
产品详情
Efalizumab 是一种靶向 T 细胞的调节剂,是 LFA-1 α 亚基 CD11a 的人源化单克隆抗体。依法珠单抗可抑制 T 细胞激活、皮肤T细胞运输和T细胞粘附到角质形成细胞,可用于斑块银屑病研究。
生物活性
Efalizumab is a targeted T cell modulator, and is a humanized monoclonal antibody of CD11a, the α subunit of LFA-1. Efalizumab inhibits T cell activation, cutaneous T cell trafficking, and T cell adhesion to keratinocytes, can be used for plaque psoriasis research.
性状
Liquid
体外研究(In Vitro)
Efalizumab (78 ng/mL-5 mg/mL) induces a leukocytosis and downregulates LFA-1 expression on T cells in the peripheral blood.
Efalizumab (78 ng/mL-5 mg/mL) downregulates plate-bound, anti-CD3-stimulated proliferation of PBMC.
has not independently confirmed the accuracy of these methods. They are for reference only.
体内研究(In Vivo)
Efalizumab shows side effects include bacterial sepsis, viral meningitis, invasive fungal disease and progressive multifocal leukoencephalopathy (PML), a brain infection caused by reactivation of latent JC virus infection.
has not independently confirmed the accuracy of these methods. They are for reference only.
运输条件
Room temperature in continental US; may vary elsewhere.
储存方式
Please store the product under the recommended conditions in the Certificate of Analysis.
ClinicalTrial
参考文献
[1]. Leonardi CL. Efalizumab: an overview. J Am Acad Dermatol. 2003 Aug;49(2 Suppl):S98-104.
[2]. Berger JR, et al. Monoclonal antibodies and progressive multifocal leukoencephalopathy. MAbs. 2009 Nov-Dec;1(6):583-9.
[3]. Koszik F, et al. Efalizumab modulates T cell function both in vivo and in vitro. J Dermatol
搜索质检报告(COA)
[1]. Leonardi CL. Efalizumab: an overview. J Am Acad Dermatol. 2003 Aug;49(2 Suppl):S98-104.
[2]. Berger JR, et al. Monoclonal antibodies and progressive multifocal leukoencephalopathy. MAbs. 2009 Nov-Dec;1(6):583-9.
[3]. Koszik F, et al. Efalizumab modulates T cell function both in vivo and in vitro. J Dermatol

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