Trimethobenzamide hydrochloride|554-92-7|(盐酸曲美苄胺; 盐酸三甲氧苯酰胺; Ro 2-9578)-陌孚医药/Medlife

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Trimethobenzamide hydrochloride (Synonyms: 盐酸曲美苄胺; 盐酸三甲氧苯酰胺; Ro 2-9578)

目录号: PL02888 纯度: ≥99%

CAS No. :554-92-7

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中文名称	Trimethobenzamide hydrochloride
中文别名	盐酸曲美苄胺;盐酸三甲氧苯酰胺;(S)-(-)-2-哌啶乙醇;盐酸曲美苄胺 USP标准品;盐酸三甲氧苯酰胺标准品;N-[4-[2-(二甲氨基)乙氧基]苄基]-3,4,5-三甲氧基苯甲酰胺盐酸盐
英文名称	Trimethobenzamide hydrochloride
英文别名	N-(4-(2-(Dimethylamino)ethoxy)benzyl)-3,4,5-trimethoxybenzamide hydrochloride;Trimethobenzamide Hydrochloride;Benzamide,N-[[4-[2-(dimethylamino)ethoxy]phenyl]methyl]-3,4,5-trimethoxy-, hydrochloride(1:1);N-[[4-[2-(dimethylamino)ethoxy]phenyl]methyl]-3,4,5-trimethoxybenzamide,hydrochloride;TRIMETHOBENZAMIDE;Trimethobenzamide Hy;3,4,5-Trimethoxy-benzoesaeure-[4-(2-dimethylamino-aethoxy)-benzylamid],Hydrochlorid;3,4,5-trimethoxy-benzoic acid-[4-(2-dimethylamino-ethoxy)-benzylamide],h;Ametik hydrochloride;N-[p-[(2-dimethylamino)ethoxy]benzyl]-3,4,5-trimethoxybenzamide hydrochloride;Nauseton;Poligerim;Tigan;trimethobenzamide chlorohydrate;trimethoxybenzamide hydrochloride;UNII-WDQ5P1SX7Q;N-{{4-[2-(Dimethylamino)ethoxy]phenyl}methyl}-3,4,5-trimethoxybenzamide monohydrochloride;N-[4-[2-(Dimethylamino)ethoxy]benzyl]-3,4,5-trimethoxybenzamide Hydrochloride;Trimethobenzamide HCL;Ibikin;Anaus;Tebamide;WDQ5P1SX7Q;Trimethobenzamide hydrochloride [USP];AK140655;Ticon;N-(p-(2-(Dimethylamino)ethoxy)benzyl)-3,4,5-trimethoxybenzamide hydrochloride;4-(2-Dimethylaminoethoxy)-N-(3,4,5-trimethoxybenzoyl)benzylamine hydrochloride;N-(p-(2-(Dimethyl;Ro 2-9578
Cas No.	554-92-7
分子式	C₂₁H₂₉ClN₂O₅
分子量	424.92
包装储存	4°C, sealed storage, away from moistur In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

产品详情

Trimethobenzamide hydrochloride 是多巴胺 D₂ 受体阻断剂，可用作预防恶心和呕吐的止吐剂。

生物活性

Trimethobenzamide hydrochloride is a blocker of the D 2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.

性状

Solid

IC50 & Target[1][2]

D2 receptor

体外研究(In Vitro)

Trimethobenzamide is a (non-phenothiazine) benzamide antiemetic that acts centrally to block D2 receptors, thereby inhibiting the medullary chemoreceptor trigger zone by blocking emetic impulses to the vomiting center. has not independently confirmed the accuracy of these methods. They are for reference only.

体内研究(In Vivo)

The oral bioavailability of Trimethobenzamide is 60% to 100%. The time to peak is about 45 minutes after oral administration and; Intramuscular (I.M.) administration about 30 minutes after intramuscular administration. has not independently confirmed the accuracy of these methods. They are for reference only.

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

4°C, sealed storage, away from moistur In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

ClinicalTrial

参考文献

[1]. Smith HS, et al. Dopamine receptor antagonists. Ann Palliat Med. 2012 Jul;1(2):137-42.

溶解度数据	In Vitro: DMSO : ≥ 100 mg/mL (235.34 mM)配制储备液

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产品使用指南

Data Sheet

1：一般建议：溶解度为Medlife测试数据，可能与文献描述存在差异。这是由于生产工艺和批次不同产生的正常现象。为了使其更好的溶解，请用37℃加热试管并在超声波水浴中震动片刻。不同批次产品溶解度各有差异，仅做参考，具体以实验方案为准。

2：储存条件：粉末-20°C一般情况可以保存3年，溶于溶剂-80°C一般情况可以保存1年。不同产品及不同批次产品可能存在差异，请细致阅读产品信息，并辅助参考相关文献描述。

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