| PL03609 |
XMU-MP-3
|
XMU-MP-3 是一种有效的非共价 BTK 抑制剂,在 10 μM ATP 存在下,对 BTK WT 和 BTK C481S 突变型的 IC50 分别为 10.7 nM 和 17.0 nM。XMU-MP-3 也诱导凋亡 (apoptosis)。 |
≥98% |
| PC30313 |
hsa-miR-4720-5p 模拟物
|
hsa-miR-4720-5p mimic 是一种化学合成的miRNA模拟物,能模拟内源性miRNA,上调miRNA活性,用于功能获得性(gain-of-function)研究。 |
|
| PL04233 |
SOP1812
|
SOP1812 是一种 naphthalene diimide (ND) 衍生物,具有抗肿瘤活性。SOP1812 能够与quadruplex arrangements (G4s) 结合,并下调多个癌症基因通路。SOP1812 对 hTERT G4 和 HuTel21 具有很强的亲和力,其 KD 值分别为 4.9 和 28.4 nM。G4SOP1812 可用于癌症的研究。 |
≥98% |
| PC57468 |
Doxepin N-oxide (hydrate)
|
Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Product Type|Biochemicals|Transporter & Exchanger Modulators||Product Type|Biochemicals|Xenobiotic Metabolites||Research Area|Neuroscience|Behavioral Neuroscience|Depression||Research Area|Neuroscience|Behavioral Neuroscience|Sleep & Biological Rhythms||Research Area|Neuroscience|Pain Research||Research Area|Toxicology & Xenobiotic Metabolism|Drug Metabolites |
|
| PC83380 |
牛蒡子醇 B
|
|
HPLC≥98% |
| PC81220 |
乌来糖
|
|
GC≥98% |
| PC54346 |
15-epi Prostaglandin A1
|
Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |
≥95% |
| PC55453 |
Doxorubicinol (hydrochloride)
|
Product Type|Biochemicals|Antibiotics|Anthracyclines||Product Type|Biochemicals|Small Molecule Inhibitors|ATPases||Product Type|Biochemicals|Small Molecule Inhibitors|Topoisomerases||Product Type|Biochemicals|Transporter & Exchanger Modulators||Product Type|Biochemicals|Xenobiotic Metabolites||Research Area|Cancer|Cell Death|Apoptosis||Research Area|Cancer|Cell Signaling|p53 Signaling||Research Area|Cancer|DNA Damage and Repair|DNA Intercalating Agents||Research Area|Cancer|DNA Damage and Repair|Topoisomerase||Research Area|Cancer|Immunology||Research Area|Cancer|Transcription Factors|p53||Research Area|Cancer|Tumor Microenvironment||Research Area|Cardiovascular System|Heart|Myocardial Contractility||Research Area|Toxicology & Xenobiotic Metabolism|Drug Metabolites||Research Area|Toxicology & Xenobiotic Metabolism|Organ- & System-Specific Toxicity|Cardiovascular |
≥90%(mixtureofisomers) |
| PC75318 |
弗罗利辛二水合物
|
植物来源:海棠叶Malus、Chaenomeles,苹果树枝叶Malus pumila Mill.; |
≥98% |
| PL05444 |
Mangafodipir trisodium
|
Mangafodipir trisodium (MnDPDP) 是肝细胞特异性造影剂,也是一种有效的 CIPN (化疗诱导的周围神经通路)和其他细胞氧化应激引起的条件抑制剂。Mangafodipir trisodium 对化疗的肿瘤杀伤活性无负干扰。 |
≥99% |