有许多抑制剂、激动剂和拮抗剂我们无法进行精确分类,因为研究领域仍然未知。
| 货号 | 产品名 | Cas | 产品描述 |
|---|---|---|---|
| PC15951 | ZIP (SCRAMBLED) | 908012-18-0 | PKMζ抑制剂,ZIP(Scrambled) 是一种杂乱肽,可用作 zeta 抑制肽 (ZIP) 的阴性对照。 |
| PC10492 | ZK 164015 | 177583-70-9 | 雌激素受体沉默拮抗剂 |
| PC11253 | ZK 756326 | 874911-96-3 | CCR8趋化因子受体激动剂,ZK756326 is a full agonist of CCR8(Chemokine receptor 8) with an IC50 of 1.8 μM, dose-responsively eliciting an increase in intracellular calcium and cross-desensitizing the response of the receptor to CCL1 |
| PC12242 | ZK 93423 hydrochloride | 1216574-52-5 | GABAA受体激动剂,ZK-93423是来自β咔啉家族的一种抗焦虑药,是一种非苯二氮卓类 GABAA受体激动剂。GABAA受体是一种配体门控离子通道和离子型受体。 |
| PC17717 | ZK118182 isopropyl ester(solution) | 154927-31-8 | ZK118182 isopropyl ester |
| PC14690 | ZLJ-6 | 1051931-39-5 | COX和5-脂氧合酶(5-LO)的双重抑制剂 |
| PC12141 | ZM 226600 | 147695-92-9 | Kir6(KATP)通道开放剂 |
| PC10086 | ZM 449829 | 4452-06-6 | JAK3抑制剂,ZM 449829 是有效的、选择性和ATP竞争性的 JAK3 抑制剂,pIC50 值为 6.8。ZM 449829 是可用于研究 JAK3 的药理学工具。 |
| PC12296 | Zoniporide dihydrochloride | 241799-10-0 | 钠氢交换异构体1(NHE1)抑制剂 |
| PC17458 | α-(difluoromethyl)-DL-Arginine | 69955-43-7 | α-(difluoromethyl)-DL-Arginine |
| PC17781 | α-CEHC | 4072-32-6 | α-CEHC |
| PC18289 | α-D-Galactopyranosylphenyl isothiocyanate | 120967-92-2 | α-D-Galactopyranosylphenyl isothiocyanate |
| PC18870 | α-D-Glucose-1,6-biphosphate (cyclohexyl ammonium salt hydrate) | 71662-13-0 | α-D-Glucose-1,6-biphosphate (cyclohexyl ammonium salt hydrate) |
| PC15406 | α-Guanidinoglutaric Acid | 73477-53-9 | nNOS的线性混合型抑制剂 |
| PC13642 | α-hederin | 27013-91-8 | alpha-hederin是能够水溶的五环三萜皂苷,有很多化学特性,例如止痉挛,驱虫,和抑制细胞增长。 |
| PC18262 | α-hydroxy Farnesyl Phosphonic Acid | 148796-53-6 | α-hydroxy Farnesyl Phosphonic Acid |
| PC18483 | α-Linolenoyl Ethanolamide(solution) | 57086-93-8 | α-Linolenoyl Ethanolamide |
| PC11059 | α-Methyl-5-hydroxytryptamine maleate | 97469-12-0 | 5-HT2B受体激动剂,α-methyl Serotonin (maleate) is an agonist of serotonin (5-HT) receptors |
| PC17546 | α-Phenyl-α-(2-pyridyl)acetonitrile | 5005-36-7 | MCC950 是一种有效的选择性NLRP3 抑制剂,作用于BMDMs 和 HMDMs,IC50 分别为 7.5 nM 和 8.1 nM。 |
| PC12117 | β-CCB | 84454-35-3 | 苯并二氮杂受体的配体 |
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