Bunazosin is a potent and selective α1-adrenoceptor antagonist. Bunazosin can be used for antihypertensive and ocular hypotensive research.
性状
Solid
IC50 & Target[1][2]
α1-adrenergic receptor
运输条件
Room temperature in continental US; may vary elsewhere.
储存方式
Powder -20°C 3 years;4°C 2 years
ClinicalTrial
参考文献
[1]. Hideaki Hara , et al. Bunazosin, a selective alpha1-adrenoceptor antagonist, as an anti-glaucoma drug: effects on ocular circulation and retinal neuronal damage. Cardiovasc Drug Rev. Spring 2005;23(1):43-56.
溶解度数据
In Vitro: DMSO : 100 mg/mL (267.77 mM; Need ultrasonic)配制储备液
[1]. Hideaki Hara , et al. Bunazosin, a selective alpha1-adrenoceptor antagonist, as an anti-glaucoma drug: effects on ocular circulation and retinal neuronal damage. Cardiovasc Drug Rev. Spring 2005;23(1):43-56.