| PL04233 |
SOP1812
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SOP1812 是一种 naphthalene diimide (ND) 衍生物,具有抗肿瘤活性。SOP1812 能够与quadruplex arrangements (G4s) 结合,并下调多个癌症基因通路。SOP1812 对 hTERT G4 和 HuTel21 具有很强的亲和力,其 KD 值分别为 4.9 和 28.4 nM。G4SOP1812 可用于癌症的研究。 |
≥98% |
| PC57468 |
Doxepin N-oxide (hydrate)
|
Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Product Type|Biochemicals|Transporter & Exchanger Modulators||Product Type|Biochemicals|Xenobiotic Metabolites||Research Area|Neuroscience|Behavioral Neuroscience|Depression||Research Area|Neuroscience|Behavioral Neuroscience|Sleep & Biological Rhythms||Research Area|Neuroscience|Pain Research||Research Area|Toxicology & Xenobiotic Metabolism|Drug Metabolites |
|
| PC83380 |
牛蒡子醇 B
|
|
HPLC≥98% |
| PC81220 |
乌来糖
|
|
GC≥98% |
| PC54346 |
15-epi Prostaglandin A1
|
Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway |
≥95% |
| PC55453 |
Doxorubicinol (hydrochloride)
|
Product Type|Biochemicals|Antibiotics|Anthracyclines||Product Type|Biochemicals|Small Molecule Inhibitors|ATPases||Product Type|Biochemicals|Small Molecule Inhibitors|Topoisomerases||Product Type|Biochemicals|Transporter & Exchanger Modulators||Product Type|Biochemicals|Xenobiotic Metabolites||Research Area|Cancer|Cell Death|Apoptosis||Research Area|Cancer|Cell Signaling|p53 Signaling||Research Area|Cancer|DNA Damage and Repair|DNA Intercalating Agents||Research Area|Cancer|DNA Damage and Repair|Topoisomerase||Research Area|Cancer|Immunology||Research Area|Cancer|Transcription Factors|p53||Research Area|Cancer|Tumor Microenvironment||Research Area|Cardiovascular System|Heart|Myocardial Contractility||Research Area|Toxicology & Xenobiotic Metabolism|Drug Metabolites||Research Area|Toxicology & Xenobiotic Metabolism|Organ- & System-Specific Toxicity|Cardiovascular |
≥90%(mixtureofisomers) |
| PC75318 |
弗罗利辛二水合物
|
植物来源:海棠叶Malus、Chaenomeles,苹果树枝叶Malus pumila Mill.; |
≥98% |
| PL05444 |
Mangafodipir trisodium
|
Mangafodipir trisodium (MnDPDP) 是肝细胞特异性造影剂,也是一种有效的 CIPN (化疗诱导的周围神经通路)和其他细胞氧化应激引起的条件抑制剂。Mangafodipir trisodium 对化疗的肿瘤杀伤活性无负干扰。 |
≥99% |
| PL05132 |
Galanthamine-O-methyl-d3
|
Galanthamine-O-methyl-d3 是 Galanthamine 的氘代物。Galanthamine 是一种有效的乙酰胆碱酯酶 (AChE) 抑制剂,IC50 为 500 nM。 |
|
| PL02692 |
TBK1/IKKε-IN-4
|
TBK1/IKKε-IN-4 是一种 6-氨基吡唑并嘧啶衍生物,也是一种有效的,选择性的 TBK1 和 IKKε 抑制剂,IC50 值分别为 13 nM 和 59 nM。TBK1/IKKε-IN-4 对其他蛋白质激酶(包括 PDK1,PI3K 家族成员和 mTOR)的活性降低了 100-1000 倍。 |
≥99% |